Intestine

Intestine
Human TransportersGenePortaCellTecITC/FDAEMAPMDA
MDR1 (P-gp)ABCB1yes+++
BCRPABCG2yes+++
MRP2ABCC2yes−−−
MRP3ABCC3yes−−−
OCT1SLC22A1yesconsider+−
ASBTSLC10A2yes−−−
PEPT1SLC15A1yes−−−
PEPT2SLC15A2yes−−−
OATP2B1SLCO2B1yes−−−
OATP2A1SLCO2A1yes−−−
NaDC1SLC13A2yes−−−
THTR1SLC19A2upon request−−−
THTR2SLC19A3upon request−−−
ENT1SLC29A1upon request−−−
ENT2SLC29A2upon request−−−
MCT1SLC16A1upon request−−−
OSTα/βSLC51A/SLC51Byes−−−
SGLT1

SLC5A1
yes

➦ Upon request we are able to stably overexpress each membrane transporter protein into HEK293 cell line.